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trons surround atoms more or less uniformly,

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Information about Using Technology to Study Cellular and Molecular Biology

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Using Technology to Study Cellular and Molecular Biology

Figure 12. The X-ray crystallography process.

it is possible to determine where atoms are

One of the most striking advancements has

located by looking at these maps. By rotating

been the use of synchrotron X-rays, which are

the crystal and generating an electron density

produced by the bending of particle beams gen-

map for each angle of rotation, it is possible to

erated by large accelerators. In a synchrotron,

produce a three-dimensional model of the mol-

charged particles, such as electrons or posi-

ecule. If the amino acid sequence of a protein

trons, are orbited around a path nearly a mile

is known, an accurate model of the protein can

in circumference, which must be maintained

be generated by fitting the atoms of the known

in a vacuum. Understandably, synchrotrons are

sequence into the electron density map.

quite expensive to build and to maintain, and

Figure 13 shows a typical diffraction pattern for

a single orientation of a protein crystal through

which an X-ray beam has been passed. Note

the different positions and intensities of the

spots, which mark the locations where scattered

X-rays have struck the detector. The image is

divided into quadrants because the detector was

composed of four separate, adjacent modules.

The white circle to the right of center with the

white line extending to the left is a shadow

resulting from a “beamstop.” The beamstop is a

small piece of lead mounted on a metal arm. It

prevents the intense beam of unscattered X-rays

from impinging on and damaging the detector.

Figure 14 shows a three-dimensional model of a

protein that was crystallized and then analyzed

by X-ray crystallography.

Figure 13. A typical X-ray−diffraction pattern for

a single orientation of a protein crystal through

Equipment used in X-ray crystallography con-

which an X-ray beam has been passed.

tinues to undergo development and refinement.

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synchrotron radiation. A modern synchrotron

source can reduce total data collection to just

30 minutes, as compared with weeks using ear-

lier X-ray–diffraction equipment.

Determining structures by X-ray diffraction

continues to add to our understanding of DNA

replication and protein synthesis. For example,

scientists recently studied the crystal structures

of a bacterial DNA polymerase I that had DNA

primer templates bound to its active site.13

The enzyme was catalytically active, which

allowed for direct observation of the products

of several rounds of nucleotide incorporation.

The polymerase was able to retain its ability to

Figure 14. Three-dimensional structure of the

distinguish between correctly and incorrectly

DNA-repair protein MutY as determined by X-ray

paired nucleotides in the crystal. By comparing

crystallography. Graphic was produced from infor-

the structures of successive complexes, it was

mation available at http://www.rcsb.org/pdb/ .

possible to determine the structural basis for

sequence-independent recognition of correctly

formed base pairs.13

there are fewer than 20 in the world. Because

synchrotron X-ray beams are many orders of

Ribosomes are the largest asymmetric structures

magnitude brighter than the usual laboratory X-

to be solved by X-ray crystallography so far.

ray sources, data for single crystal orientations

Results, with resolutions as high as 2.4 Å, have

can be collected with exposures of a minute or

helped establish the locations of the 27 proteins

less, rather than exposures of several minutes to

and the 2,833 bases of ribosomal (rRNA) found

an hour.

within the ribosome.4 The structure also shows

that contacts between the two ribosome sub-

The completion of the Human Genome Proj-

units are limited, which helps explain why the

ect has provided the foundation for explosive

ribosome subunits dissociate so readily.

growth in structural biology. Technological

advances in X-ray crystallography have greatly

Some biomolecules or biomolecular complexes

reduced the time and effort required to solve

are not suitable for diffraction analysis because

structures. In addition to synchrotron X-

they cannot be crystallized. Scientists, however,

rays, advances include faster X-ray detectors,

are optimistic about developing techniques to

improved computational methods for process-

deal effectively with noncrystalline materials.18

ing data, and robotics for growing and handling

This will make it possible to image everything

crystals. Structure determinations that used to

from cells to individual protein molecules.

involve a 20-person, yearlong effort now con-

stitute a single chapter in a graduate student’s

4.3 Nuclear magnetic resonance (NMR)

thesis. The Protein Structure Initiative, remi-

spectroscopy

niscent of the Human Genome Project, aims to

Most people know of magnetic resonance imag-

produce the three-dimensional structures for

ing (MRI) as an important diagnostic tool in

the estimated 1,000 to 5,000 distinct spatial

medicine that can produce incredible images

arrangements assumed by polypeptides found

of soft tissues. Less well known is that MRI

in nature. Such high-throughput data collection

represents only a limited area of NMR. NMR

is best suited to X-ray crystallography using

depends on the fact that atomic nuclei having

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Information about Using Technology to Study Cellular and Molecular Biology

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Using Technology to Study Cellular and Molecular Biology

an odd number of protons, neutrons, or both

in plants. This enzyme functions as a molecular

have an intrinsic spin. When such a nucleus is

motor that uses an internal rotary mechanism.

placed in a magnetic field, it can align either in

NMR has been used to reveal structural changes

the same direction as the field or in the oppo-

in a protein subunit of the enzyme that may

site direction. A nucleus aligned with the field

explain how the rotation is driven.20

has a lower energy than one aligned against it.

NMR spectroscopy refers to the absorption of

Many see the successful Human Genome Project

radiofrequency radiation by nuclei in a strong

as providing a foundation for a major initiative

magnetic field. Absorption of energy causes the

in structural biology in which NMR will play

nuclei to realign in the higher-energy direction.

a critical role.5 Informal groups of scientists in

The nuclei then emit radiation and return to

the United States are proposing the creation of

the lower-energy state. The local environment

10 regional “collaboratories,” each with power-

around each nucleus will distort the magnetic

ful new-generation NMR spectrophotometers

field slightly and affect its transition energy.

to assist with high-throughput structure deter-

This relationship between transition energy and

minations. Universities, too, are interested in

an atom’s position within a molecule allows

establishing collaborative centers in genomics

NMR to provide structural information.

and proteomics.9 At Stanford, Nobel Prize–

winning physicist Steven Chu and biochemist

One advantage of NMR spectroscopy over X-ray

James Spudich are leading an effort to create

crystallography and electron microscopy is that

an interdisciplinary research center housing 50

it can be applied to the study of movement at

faculty members, while Princeton University is

the molecular level. NMR studies are providing

planning to add an interdisciplinary genomics

a growing list of cases where conformational

institute to its molecular biology department.

dynamics correlate with protein-protein interac-

tion on surfaces. For example, the enzyme ATP

4.4 Laser technology

synthase catalyzes the formation of ATP from

When the laser made its first appearance in

ADP and phosphate during oxidative phosphor-

the 1950s, it was a tool without a task. Since

ylation in animals and photophosphorylation

then, the laser has been put to myriad uses in

our everyday lives—from scanning prices at the

supermarket to playing music and printing text.

Similarly, in scientific research, the laser has

found many applications. It is like a Swiss Army

knife, having many blades with a variety of uses.

Combining lasers and microscopy has greatly

expanded our ability to image cellular and

molecular structures. Cells, or parts of cells,

can be exposed to antibodies or nucleic acid

probes labeled with fluorescent dyes. When

excited by laser light of the appropriate wave-

length, specific areas of the cell, or regions of

a chromosome, can be visualized. The resolu-

tion of optical microscopy is limited by physical

laws. Diffraction prevents the laser beam (and

therefore the spot of fluorescence) from being

focused any finer than about 200 nm. However,

a new approach is overcoming this limit. It uses

Figure 15. Equipment for high-resolution nuclear

a combination of two laser beams, one to illu-

magnetic resonance (NMR) spectroscopy.

minate and image the sample, and a second that

34

shapes the first beam and reduces the effects of

diffraction. The technique has been used to dis-

The amount of genetic data available

tinguish crystals only 100 nm apart and is still

and the rate of acquisition are astonish-

undergoing improvement.

ing by any measure.

Lasers, together with magnets, are being used

to develop technologies for manipulating single

The use of computers to model protein folding

molecules. Investigators are now able to exam-

is one of the primary efforts in the postsequenc-

ine how DNA interacts with the various protein

ing phase of the Human Genome Project. In the

molecules that cut, paste, and copy it. DNA is

1970s, when the first proteins were modeled,

an ideal choice for single-molecule studies. It

the structures generated were in vacuo (in a vac-

is a very large molecule (the longest human

uum), with no other molecules interacting with

chromosome stretches to 9 centimeters) and

the protein. Of course, each protein in a living

quite robust. For example, scientists have suc-

cell is surrounded by thousands of water mol-

ceeded in using lasers as optical tweezers to tie

ecules, and these have an important effect on

knots in single DNA molecules.2 Results indi-

the protein’s conformation. Indeed, research has

cate that knotted DNA is stronger than actin, a

demonstrated that the water-containing models

major muscle protein. Although tying DNA into

of proteins are much better predictors of how

knots may not seem particularly useful, it does

the proteins look and function within a cell.10

provide insight into the molecule’s mechanical

properties, which are critical to understanding

The importance of protein folding was recently

how enzymes interact with it.

recognized by IBM, which announced that it

would spend $100 million to build a supercom-

4.5 Simulations and computations

puter called Blue Gene. The five-year IBM initia-

The explosion of data produced by the Human

tive will involve modeling how proteins take on

Genome Project led to the creation of a new

their three-dimensional shapes. A major aim is

discipline, bioinformatics, whose focus is on

to help drug researchers identify drug targets for

the acquisition, storage, analysis, modeling, and

treating diseases. Protein folding is a daunting

distribution of the many types of information

problem. Even Blue Gene, which will be 500

embedded in DNA and protein-sequence data.14

times faster than the current fastest computer,

Biologists are familiar with the terms in vivo and

will require about one year to simulate the com-

in vitro, used to describe processes that occur

plete folding of a typical protein. The stakes,

in the body and in the test tube, respectively.

however, are huge. Approximately one-third

Now they are becoming acquainted with a new

of the genes identified in the newly sequenced

term, in silico, used to describe a new branch

human genome are of unknown function and

of biology that requires little more than a com-

are therefore of particular academic and com-

puter and a connection to the Internet. As more

mercial interest. New companies are formed

and more DNA and protein sequence data find

on a monthly basis to take part in this genetics

their way into computer databases, the ability

sweepstakes.

of bioinformatics to address biological ques-

tions becomes more powerful. The amount of

5 Technology and the Origins of

genetic data available and the rate of acquisition

Molecular Biology

are astonishing by any measure. According to

This section provides a brief history of the ori-

Francis Collins, head of the National Human

gins of molecular biology. It addresses the gene’s

Genome Research Institute, it took four years

chemical nature, organization, and behavior.

to obtain the first 1 billion base pairs of human

Despite molecular biology’s narrow focus on

sequence and just four months to get the second

DNA, it is readily apparent that many of the

billion.16

most important advances in the field have relied

35

Information about Using Technology to Study Cellular and Molecular Biology Using Technology to Study Cellular and Molecular Biology

heavily on technology-based contributions from

unaware of the important one-gene–one-enzyme

chemistry and physics. This is addressed in the

work of George Beadle and Edward Tatum from

National Science Education Standards. The His-

the early 1940s), the book has been credited

tory and Nature of Science Content Standard

with influencing a generation of physicists to

G states, “As a result of activities in grades 9 to

consider biological questions.

12, all students should develop understanding

of . . . historical perspectives.” It further states,

Soon, the ranks of the Phage Group began to

“Occasionally, there are advances in science and

grow. It included other physicists, such as Leo

technology that have important and long-lasting

Szilard, holder of the patent for the nuclear

effects on science and society.”

chain reaction and a participant in the Man-

hattan Project, and Thomas Anderson, one

Science historians often attribute the origins of

of the first American electron microscopists.

molecular biology to the Phage Group, which

Micrographs obtained by Anderson and Roger

first met in 1940 at Cold Spring Harbor Labora-

Herriott showed that phage begin the infection

tory in Long Island, N.Y. At the center of the

process by attaching to bacteria by their tails.

group were three scientists. Max Delbrück, a

Later, empty phage “ghosts” could be seen on

German physicist working at Vanderbilt Uni-

the bacterial surface.

versity, and Salvador Luria, an Italian biologist

working at Indiana University, had fled to the

Hershey and his colleague Martha Chase used

United States from Nazi Europe. They were

phage to examine the molecular nature of the

joined at Cold Spring Harbor by Alfred Hershey,

gene.11 They took advantage of radioactive iso-

an American biologist working for the Carnegie

topes that became available as a consequence

Institution’s Department of Genetics.

of work on the atomic bomb. Despite the ear-

lier work of Oswald Avery and his colleagues

Bacteriophage, also called phage, are viruses

demonstrating that DNA was the hereditary

that infect bacteria.1 These were discovered in

substance,3 many scientists continued to believe

1916 by the English microbiologist F.W. Twort

that genes could only be made of protein. Her-

and, independently, two years later by the

shey and Chase began their experiment by

French-Canadian F. d’Herelle. It was d’Herelle

using radioactive phosphorous to label phage

who came up with the name bacteriophage.

DNA and radioactive sulfur to label phage pro-

Phage became an important area of research in

tein. They tried to detect which radiolabel went

the 1920s, when scientists hoped they could be

inside the bacterium to direct synthesis of new

used to treat bacterial diseases. When this hope

phage particles after the bacterium was infected.

failed to materialize, phage research fell out of

At first, they could not effectively detach the

favor until the Phage Group resurrected it.22

phage particles from the surfaces of the bacte-

rial cells, but then an unexpected technology

In 1944, Delbrück organized a summer course

came to their aid. They used a Waring blender,

at Cold Spring Harbor Laboratory to introduce

originally designed to mix cocktails, to disrupt

other scientists to the quantitative methods for

the attachments of the phage to the bacterial

studying phage that he and Luria had devel-

cells. The radioactive phosphorous went into

oped. In that same year, the great Austrian

the bacterial cells, while the radioactive sulfur

physicist Erwin Schrödinger published a book

remained outside with the phage ghosts, con-

titled What Is Life? that discussed heredity from

firming that DNA, and not protein, contains the

a physics perspective.19 Schrödinger reasoned

genetic information. This work set the stage for

that although living things obey the laws of

the contribution of the youngest member of the

physics, they also might be governed by undis-

Phage Group, James Watson.

covered physical laws. Although biologists of

that time regarded Schrödinger’s book as roman-

Watson came to the Cavendish Laboratory at

tic and a bit naive (for example, he seemed

Cambridge University in 1951, ostensibly to

36

study the three-dimensional structures of pro-

Samples of cells were removed before the switch

teins. He quickly fell in with Francis Crick, a

to the light-isotope growth medium (genera-

British physicist, who had developed an inter-

tion 1) and from the first two generations fol-

est in heredity after reading Schrödinger’s What

lowing the switch (generations 2 and 3). DNA

Is Life? The pair formed a collaboration that

samples extracted from the cell samples were

resulted two years later in the proposal of the

centrifuged through a solution of cesium chlo-

double helix model of DNA.23 Although Watson

ride that forms a density gradient during cen-

and Crick relied on model building to solve

trifugation (for 20 hours at 40,000 revolutions

DNA’s structure, they could not have succeeded

per minute). DNA molecules form a discrete

without help from two other scientists at Cam-

band at a position where their density equals

bridge, Maurice Wilkins and Rosalind Franklin.

that of the cesium chloride gradient. The DNA

Wilkins first, and then Franklin, used X-ray

samples taken from generation 1 contained a

diffraction to study the structure of DNA. In

single heavy band, since both DNA strands con-

the case of DNA fibers, the diffraction patterns

tained the 15N isotope. Samples from generation

suggested that the molecule was some type of a

2 displayed a single band of medium density,

helix with a diameter of 20 Å and a repeat of 34

since each DNA molecule consisted of one

Å. Near the end of the paper that describes the

heavy (15N) parental strand and one light (14N)

double helix, Watson and Crick included the

complementary strand. Finally, samples from

statement, “It has not escaped our notice that

generation 3 displayed bands of two different

the specific pairing we have postulated immedi-

densities. One band of medium density again

ately suggests a possible copying mechanism for

consisted of a heavy parental strand and a new

the genetic material.”

complementary light strand. A second band of

light density consisted of two strands of light

Experimental support for a copying mechanism

DNA, one an inherited light parental strand and

suggested by the double helix structure came in

the other, a new complementary light strand.

1958 from Matthew Meselson and Frank Stahl,

then working at the California Institute of Tech-

Around the time that Meselson and Stahl were

nology. In what some have called “the most

performing their experiments, Crick theorized

elegant experiment in molecular biology,”